Author(s): Akshay R. Yadav, Shrinivas K. Mohite

Email(s): akshayyadav24197@gmail.com

DOI: 10.5958/0975-4377.2020.00051.8   

Address: Akshay R. Yadav*, Dr. Shrinivas K. Mohite
Department of Pharmaceutical Chemistry, Rajarambapu College of Pharmacy, Kasegaon, Sangli, Maharashtra, India- 415404.
*Corresponding Author

Published In:   Volume - 12,      Issue - 4,     Year - 2020


ABSTRACT:
Use of ultrasound to accelerate reactions has proved to be especially effective method for achieving the green chemistry goals of waste minimization and energy requirements. Ultrasonic irradiation applications are playing an growing role in chemical processes, especially in cases where traditional methods require drastic conditions or prolonged reaction times. Taking account ultrasound and the origin of its effects on chemical reactions, a total of fourty-two studies of preparation of azoles under ultrasonic irradiation conditions are reviewed. Such reports were classified according to the number of heteroatoms present in the ring (2, 3 or 4) and each group subdivided by azole which includes the class of oxadiazole and thiazole. Research has shown in medicinal chemistry that compounds with biological activity are mostly dependent upon heterocyclic structures. Azoles and their derivatives in particular have attracted growing interest as versatile intermediates for the synthesis of biologically active compounds such as potent antitumors, antibacterial, antiviral, and antioxidants. Azoles are a broad class of 5-membered heterocyclic ring compounds with at least one nitrogen atom in their structure and one heteroatom in it. Because of the broad range of biological activities ascribed to structurally distinct azoles, the construction of this type of molecule has received considerable attention.


Cite this article:
Akshay R. Yadav, Shrinivas K. Mohite. Recent advances in the Ultrasound-Assisted synthesis of Oxadiazole and Thiazole Derivatives. Res. J. Pharma. Dosage Forms and Tech.2020; 12(4):308-312. doi: 10.5958/0975-4377.2020.00051.8

Cite(Electronic):
Akshay R. Yadav, Shrinivas K. Mohite. Recent advances in the Ultrasound-Assisted synthesis of Oxadiazole and Thiazole Derivatives. Res. J. Pharma. Dosage Forms and Tech.2020; 12(4):308-312. doi: 10.5958/0975-4377.2020.00051.8   Available on: https://rjpdft.com/AbstractView.aspx?PID=2020-12-4-13


REFERENCES:
1.    Shelke, S.; Mhaske, G.; Gadakh, S. and Gill, C. Green synthesis and biological evaluation of some novel azoles as antimicrobial agents. Bioorg Med Chem Let. 2010; 20: 7200-7204.
2.    Ahirrao, P. Recent developments in antitubercular drugs. Mini Rev. Med. Chem. 2008; 8: 1441–1451.
3.    Migliori, G.B.; DeLaco, G.; Besozzi, G.; Centis, R.; Cirillo, D.M. First tuberculosis cases in Italy resistant to all tested drugs. Euro Surveill. 2007; 12: 3194.
4.    Diacon, A.H.; Donald, P.R.; Pym, A.; Grobusch, M.; Patientia, R.F.; Mahanyele, R.; Bantubani, N.; Narasimooloo, R.; De Marez, T.; van Heeswijk, R.. Randomized pilot trial of eight weeks of bedaquiline (TMC207) treatment for multidrug-resistant tuberculosis: Long-term outcome, tolerability, and effect on emergence of drug resistance. Antimicrob. Agents Chemother. 2012; 56: 3271–3276.
5.    Yadav A, Mohite S, Design, Synthesis and Characterization of Some Novel benzamide derivatives and it’s Pharmacological Screening. 2020. Int J Sci Res Sci Technol. 7(2): 68-74.
6.    Yadav A, Mohite S, Magdum C, Synthesis, Characterization and Biological Evaluation of Some Novel 1,3,4-Oxadiazole Derivatives as Potential Anticancer Agents, Int J Sci Res Sci Technol. March-April-2020; 7 (2): 275-282.
7.    Rajput M. D, Yadav A. R, Mohite S.K, Synthesis, Characterization of Benzimidazole Derivatives as Potent Antimicrobial Agents. 2020. Int. J. Pharm. 17(4): 279-285.
8.    Shinde, A. D.; Kale, B. Y.; Shingate, B. B. andShingare, M. S. Synthesis and characterization of 1-benzofuran-2-yl thiadiazoles, triazoles and oxadiazoles by conventional and non-conventional methods. J KorChem Soc. 2010; 54: 582-588.
9.    Shinde, A. D.; Sonar, S. S.; Shingate, B. B. and Shingare, M. S. Synthesis and biological screening of novel thiadiazoles, selenadiazoles, and spirocyclicbenzopyran by ultrasonic and microwave irradiation. Phosphorus, Sulfur, and Silicon. 2010; 185: 1594-1603.
10.    Silva, F. A. N.; Galluzzi, M. P.; Albuquerque, B.; Pizzuti, L.; Gressler, V.; Rivelli, D. P.; Barros, S. B. M. and Pereira, C. M. P. Ultrasound irradiation promoted largescale preparation in aqueous media and antioxidant activity of azoles. Let Drug Design andDiscov. 2009; 6: 323-326.
11.    Tiwari, V.; Parvez, A. and Meshram. J. Benign methodology and improved synthesis of 5-(2-chloroquinolin-3-yl)-3-phenyl-4,5-dihydroisoxazoline using acetic acid aqueous solution under ultrasound irradiation. UltrasonSonochem. 2008; 18: 911-916.
12.    Venzke, D.; Flores, A. F. C.; Quina, F. H.; Pizzuti, L. and Pereira, C. M. P. Ultrasound promoted greener synthesis of 2-(3,5-diaryl-4,5-dihydro-1H-pyrazol-1-yl)-4phenylthiazoles. UltrasonSonochem. 2009; 18: 370-374.
13.    Yuan, Y.-Q. and Guo, S.-R. TMSCl/Fe (NO3)3-Catalyzed synthesis of 2arylbenzothiazoles and 2-arylbenzimidazoles under ultrasonic irradiation. SynCommun. 2011; 41: 2169-2177.
14.    Zang, H.; Su, Q.; Mo, Y.; Cheng, B.-W. and Jun, S. Ionic liquid [emim]OAc under ultrasonic irradiation towards the first synthesis of trisubstitutedimidazoles. UltrasonSonochem. 2010; 17: 749-751.
15.    Pizzuti, L.; Martins, P. L. G.; Ribeiro, B. A.; Quina, F. H.; Pinto, E.; Flores, A. F. C.; Venzke, D. and Pereira, C. M. P. Efficient sonochemical synthesis of novel 3,5-diaryl4,5-dihydro-1H-pyrazole-1-carboximidamides. UltrasonSonochem, 2010; 17: 34-37.
16.    Pizzuti, L.; Piovesan, L. A.; Flores, A. F. C.; Quina, F. H. and Pereira, C. M. P. Environmentally friendly sonocatalysis promoted preparation of 1-thiocarbamoyl3,5-diaryl-4,5-dihydro-1H-pyrazoles. UltrasonSonochem. 2009; 16: 728-731.
17.    Richards, W. T. and Loomis, A. L. The chemical effects of high-frequency sound waves. I. A preliminary survey. Journal of the American Chemical Society. 1927; 49: 30863100.
18.    Rodrigues-Santos, C. E. and Echevarria, A. (2011). Convenient syntheses of pyrazolo [3,4b] pyridin-6-ones using either microwave or ultrasound irradiation. Tetrahedron Let. 2010; 52: 336-340.
19.    Saleh, T. S. and El-Rahman, T. S. Ultrasound promoted synthesis of substituted pyrazoles and isoxazoles containing sulphone moiety. UltrasonicsSonochemistry, 2009; 16: 237-242.
20.    Sant’Anna, G. S.; Machado, P.; Sauzem, P. D.; Rosa, F. A.; Rubin, M. A.; Ferreira, J.; Bonacorso, H. G.; Zanatta, N. and Martins, M. A. P. Ultrasound promoted synthesis of 2-imidazolines in water: a greener approach toward monoamine oxidase inhibitors. Bioorg MedChem Let. 2009; 19: 546-549.
21.    Shekouhy, M. and Hasaninejad, A. Ultrasound-promoted catalyst-free one pot four component synthesis of 2H-indazolo [2,1-b] phthalazine-triones in neutral ionic liquid 1-butyl-3-methylimidazolium bromide. UltrasonSonochem. 2010; 19: 307-313.
22.    Cravotto, G.; Cintas, P. Power ultrasound in organic synthesis: Moving cavitational chemistry from academia to innovative and large-scale applications. J. Chem. Soc. 2006, 35, 180–196.

Recomonded Articles:

Author(s): Namdeo G. Shinde, Nayana V. Pimpodkar

DOI: 10.5958/0975-4377.2015.00011.7         Access: Open Access Read More

Research Journal of Pharmaceutical Dosage Forms and Technology (RJPDFT) is an international, peer-reviewed journal, devoted to pharmaceutical sciences. ...... Read more >>>

RNI: Not Available                     
DOI: 10.5958/0975-4377 


Recent Articles




Tags